Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5AYG
TargetNuclear receptor ROR-gamma(Mouse)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153606(CHEMBL3775900)
Affinity DataEC50:  300nMAssay Description:Inhibition of mouse RORgamma ligand binding domain (Isoleucine 251 to Lysine 516) expressed in CHOK1 cells incubated for 2 days by Gal4 luciferase re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor ROR-gamma(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50153606(CHEMBL3775900)
Affinity DataEC50:  820nMAssay Description:Inhibition of human RORgamma ligand binding domain (Serine 253 to Lysine 518 residues) expressed in CHOK1 cells incubated for 2 days by Gal4 lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)