Report error Found 2 Enz. Inhib. hit(s) for PDB: 5CYI
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of South Australia Cancer Research Institute
Curated by ChEMBL
University of South Australia Cancer Research Institute
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human recombinant CDK2/untagged Cyclin A2 (174 to 432 residues) using GST-tagged pRB as substrate preincubated overnight followed by 8 ...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of South Australia Cancer Research Institute
Curated by ChEMBL
University of South Australia Cancer Research Institute
Curated by ChEMBL
Affinity DataKd: 720nMAssay Description:Binding affinity to recombinant human CDK2/CyclinA by SPR assayMore data for this Ligand-Target Pair

3D Structure (crystal)