Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5CYI
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM50511927(CHEMBL4517803)
Affinity DataIC50: 160nMAssay Description:Inhibition of human recombinant CDK2/untagged Cyclin A2 (174 to 432 residues) using GST-tagged pRB as substrate preincubated overnight followed by 8 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM50511927(CHEMBL4517803)
Affinity DataKd:  720nMAssay Description:Binding affinity to recombinant human CDK2/CyclinA by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)