Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5D7X
TargetPeregrin(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172107(CHEMBL3810303)
Affinity DataKd:  1.50E+4nMAssay Description:Competitive binding affinity to human His-tagged BRPF1b (626 to 740 residues) expressed in T7 phage-infected Escherichia coli BL21(DE3) cells measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50172107(CHEMBL3810303)
Affinity DataKd:  1.50E+4nMAssay Description:Binding affinity to recombinant GST-tagged human BRPF1 expressed in Escherichia coli BL21 (DE3) after 1 hr by qPCR-based BromoScan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)