Report error Found 25 Enz. Inhib. hit(s) for PDB: 5DH3
Affinity DataIC50: 9.80nMAssay Description:Inhibition of MST1 (unknown origin) in presence of ATP by enzymatic assayMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKd: 11nMAssay Description:Binding affinity to MST2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Binding affinity to MST1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of MST2 (unknown origin) in presence of ATP by enzymatic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant His-tagged full-length MST2 (unknown origin) expressing in Escherichia coli assessed as MOB1a phosphorylation level incubat...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of recombinant His-tagged full-length MST2 (unknown origin) expressing in Escherichia coli assessed as GST-tagged MOB1a phosphorylation le...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of Flag-tagged full-length MST2 (unknown origin) transfected in HEK293T cells assessed as MOB1a phosphorylation level incubated for 3 hrs ...More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant His-tagged full-length MST2 (unknown origin) expressing in Escherichia coli assessed as MOB1 phosphorylation level incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Inhibition of Flag-tagged full-length MST1 (unknown origin) transfected in HEK293T cells assessed as MOB1a phosphorylation level incubated for 3 hrs ...More data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Inhibition of recombinant His-tagged full-length MST1 (unknown origin) expressing in Escherichia coli assessed as MOB1 phosphorylation level incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 104nMAssay Description:Inhibition of recombinant full length N-terminal GST -tagged human MST1 expressed in baculovirus infected Sf9 insect cells using KKSRGDYMTMQIG as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 162nMAssay Description:Inhibition of MST1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 164nMAssay Description:Inhibition of recombinant His-tagged full-length MST1 (unknown origin) expressing in Escherichia coli assessed as MOB1a phosphorylation level incubat...More data for this Ligand-Target Pair
Affinity DataIC50: 177nMAssay Description:Inhibition of recombinant His-tagged full-length MST2 (unknown origin) expressing in Escherichia coli assessed as MOB1a phosphorylation level incubat...More data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant His-tagged full-length MST2 (unknown origin) expressing in Escherichia coli assessed as MOB1a phosphorylation level incubat...More data for this Ligand-Target Pair
Affinity DataIC50: 361nMAssay Description:Inhibition of recombinant His-tagged full-length MST2 Y101F mutant (unknown origin) expressing in Escherichia coli assessed as MOB1 phosphorylation l...More data for this Ligand-Target Pair
Affinity DataIC50: 378nMAssay Description:Inhibition of recombinant His-tagged full-length MST1 (unknown origin) expressing in Escherichia coli assessed as MOB1a phosphorylation level incubat...More data for this Ligand-Target Pair
Affinity DataIC50: 493nMAssay Description:Inhibition of MST2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of recombinant His-tagged full-length MST2 D109A mutant (unknown origin) expressing in Escherichia coli assessed as MOB1 phosphorylation l...More data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+3nMAssay Description:Displacement of K5 tracer from full length C-terminal NanoLuc fused human STK4 expressed in HEK293T cells incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of recombinant His-tagged full-length MST1 (unknown origin) expressing in Escherichia coli assessed as MOB1a phosphorylation level incubat...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant His-tagged full-length MST2 (unknown origin) expressing in Escherichia coli assessed as MOB1a phosphorylation level incubat...More data for this Ligand-Target Pair
Affinity DataIC50: 1.51E+3nMAssay Description:Displacement of K5 tracer from full length C-terminal NanoLuc fused human STK3 expressed in HEK293T cells incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of recombinant His-tagged full-length MST2 Y101F/D109A mutant (unknown origin) expressing in Escherichia coli assessed as MOB1 phosphoryla...More data for this Ligand-Target Pair
Affinity DataIC50: 4.04E+3nMAssay Description:Inhibition of recombinant His-tagged full-length MST1 (unknown origin) expressing in Escherichia coli assessed as MOB1a phosphorylation level incubat...More data for this Ligand-Target Pair