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Found
1
Enz. Inhib. hit(s) for PDB:
5FNQ
Target
Kelch-like ECH-associated protein 1
(Human)
Astex Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50180854
(CHEMBL3819037)
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Affinity Data
IC50: 1.00E+6nM
Assay Description:
Displacement of 5'-TAMRA-NRF2 peptide from human recombinant N-terminal His6 and Avi-tagged KEAP1 (321 to 609 residues) expressed in baculovirus infe...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
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Ligand Info
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In Depth
Date in BDB:
9/22/2017
Entry Details
Article
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PubMed
PDB
3D Structure (crystal)
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