Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 5H17
TargetPolycomb protein EED(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50259910(CHEMBL4097892)
Affinity DataIC50: 890nMAssay Description:Binding affinity to his tagged EED (1 to 441 residues) (unknown origin) incubated for 20 mins in presence of biotinylated H3K27me3 peptide (19 to 33 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPolycomb protein EED(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50259910(CHEMBL4097892)
Affinity DataIC50: 890nMAssay Description:Binding affinity to his tagged EED (1 to 441 residues) (unknown origin) incubated for 20 mins in presence of biotinylated H3K27me3 peptide (19 to 33 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPolycomb protein EED(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50259910(CHEMBL4097892)
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity to human methionine-13Cepsilon-methyl labeled PRC2-EED (76 to 441 residues) expressed in Escherichia coli BL21 (DE3) by 2D NMR metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)