Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5I83
TargetCREB-binding protein(Human)
Genentech

US Patent
LigandPNGBDBM50178192(CHEMBL3814772 | US10206931, Example 123)
Affinity DataIC50: 652nMAssay Description:His/Flag epitope tagged CBP was cloned, expressed, and purified to homogeneity. CBP binding and inhibition was assessed by monitoring the engagement ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
Genentech

US Patent
LigandPNGBDBM50178192(CHEMBL3814772 | US10206931, Example 123)
Affinity DataIC50: 4.10E+3nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP (unknown origin) incubated for 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/17/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)