Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5I8P
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50162136(CHEMBL3792924)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant human Lp-PLA2 using 2-thio-PAF as substrate measured for 10 mins by plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPlatelet-activating factor acetylhydrolase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50162136(CHEMBL3792924)
Affinity DataKd:  185nMAssay Description:Binding affinity to human Lp-PLA2 by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)