Report error Found 1 Enz. Inhib. hit(s) for PDB: 5J9L
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of full length recombinant human GST-tagged TAK1 expressed in baculovirus expression system after 1 hr by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair

3D Structure (crystal)