Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 5K0H
TargetCoagulation factor X(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50462575(CHEMBL4238121)
Affinity DataKi:  29nMAssay Description:Inhibition of human factor 10a using Boc-Leu-Gly-Arg-AMC as fluorogenic substrate measured after 10 mins by spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCoagulation factor X(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50462575(CHEMBL4238121)
Affinity DataKi:  29nMAssay Description:Inhibition of factor 10a (unknown origin) pre-incubated for 2 hrs before fluorescence substrate addition and measured after 5 mins by fluorescence as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCoagulation factor X(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50462575(CHEMBL4238121)
Affinity DataKi:  29nMAssay Description:Inhibition human FA10a using Boc-LeuGly-Arg-AMC fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)