Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5KBQ
TargetSerine/threonine-protein kinase PAK 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340555((4-methyl-3-(methyl(2-(3-(methylsulfonyl)-5-morpho...)
Affinity DataIC50: 100nMAssay Description:Inhibition of PAK1 (unknown origin) by ATP-kinaseGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PAK 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50340555((4-methyl-3-(methyl(2-(3-(methylsulfonyl)-5-morpho...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of PAK1 phosphorylation in human MCF10A cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)