Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 5LVQ
TargetHistone acetyltransferase KAT2B(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50207717(CHEMBL3110243)
Affinity DataKd:  7.30E+4nMAssay Description:Binding affinity to human His6-tagged PCAF expressed in Escherichia coli BL21(DE3)-R3 using methanol by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone acetyltransferase KAT2B(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50207717(CHEMBL3110243)
Affinity DataKd:  1.04E+5nMAssay Description:Binding affinity to human His6-tagged PCAF expressed in Escherichia coli BL21(DE3)-R3 using 0.5% DMSO by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone acetyltransferase KAT2B(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50207717(CHEMBL3110243)
Affinity DataKd:  1.66E+5nMAssay Description:Binding affinity to human His6-tagged PCAF expressed in Escherichia coli BL21(DE3)-R3 using 1% DMSO by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone acetyltransferase KAT2B(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50207717(CHEMBL3110243)
Affinity DataKd:  4.59E+5nMAssay Description:Binding affinity to human His6-tagged PCAF expressed in Escherichia coli BL21(DE3)-R3 using 3% DMSO by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)