Report error Found 2 Enz. Inhib. hit(s) for PDB: 5M96
Affinity DataIC50: 13nMAssay Description:Inverse agonist activity at His-tagged human RORgammat LBD assessed as inhibition of biotinylated RIP140 co-activator peptide binding incubated for 1...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inverse agonist activity at His tagged human RORgammat incubated for 1 hrs in presence of biotinylated co-activator peptide by FRET assayMore data for this Ligand-Target Pair

3D Structure (crystal)