Report error Found 6 Enz. Inhib. hit(s) for PDB: 5MG2
Affinity DataKd: 9.30nMAssay Description:Binding affinity to human TAF1 tandem bromodomain (1373 to 1499 residues) transfected in Escherichia coli BL21 (DE3) assessed as dissociation constan...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human TAF1 (D1521 to D1656 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Affinity DataKd: 47nMAssay Description:Binding affinity to human TAF1 BD 2 (1501 to 1635 residues) transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant by isotherma...More data for this Ligand-Target Pair
Affinity DataEC50: 70nMAssay Description:Binding affinity to TAF1 in HEK293T cells assessed as increase in TAF1 level by ITDR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 2.10E+3nMAssay Description:Binding affinity to human TAF1 tandem bromodomain (1373 to 1499 residues) transfected in Escherichia coli BL21 (DE3) assessed as dissociation constan...More data for this Ligand-Target Pair
Affinity DataKd: 4.60E+3nMAssay Description:Binding affinity to human TAF1 BD 1 (1373 to 1499 residues) transfected in Escherichia coli BL21 (DE3) by isothermal titration calorimetric analysisMore data for this Ligand-Target Pair