Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5O4S
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50468537(CHEMBL4286098)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to N-terminal GST-tagged BRPF1 (unknown origin) expressed in Escherichia coli by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50468537(CHEMBL4286098)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)