Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5SJL
LigandPNGBDBM120470(US8703768, 70 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 2.08nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM120470(US8703768, 70 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 2.10nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)