Report error Found 6 Enz. Inhib. hit(s) for PDB: 5T3Q
Affinity DataKi: 2.70nMAssay Description:Inhibition of c-Met by HTRF assayMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 2.70nMAssay Description:Inhibition of human c-METMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nM ΔG°: -48.4kJ/molepH: 7.4 T: 2°CAssay Description:In vitro kinase assays were done to establish IC50 values against recombinant enzymes using homogeneous time-resolved fluorescence (HTRF) assay. For ...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of MET (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of c-Met (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of HGF-mediated c-Met autophosphorylation in human PC3 cells after 10 mins by quantitative electrochemiluminescent immunoassayMore data for this Ligand-Target Pair