Report error Found 6 Enz. Inhib. hit(s) for PDB: 5T8E
Affinity DataEC50: 0.190nMAssay Description:Agonist activity at human AR expressed in African green monkey COS7 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.190nMAssay Description:Modulation of Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Agonist activity at androgen receptor (unknown origin) expressed in African green monkey COS7 cells after 24 hrs by MMTV-promoter driven luciferase r...More data for this Ligand-Target Pair
Affinity DataIC50: 0.720nMAssay Description:Inhibition of Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.720nMAssay Description:Displacement of [17-alpha-methyl-H-3] mibolerone from wild-type androgen receptor (unknown origin) expressed in Freestyle293F cells measured after 3 ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.720nMAssay Description:Displacement of [3H]mibolerone from human AR after 3 hrsMore data for this Ligand-Target Pair

3D Structure (crystal)