Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 5ULA
TargetBromodomain-containing protein 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591847(CHEMBL5194033)
Affinity DataKi:  77nMAssay Description:Binding affinity to human BRD4 BD1 assessed as inhibition constant incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591847(CHEMBL5194033)
Affinity DataKi:  77nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) by a fluorescence anisotropy binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591847(CHEMBL5194033)
Affinity DataKi:  718nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) by a fluorescence anisotropy binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591847(CHEMBL5194033)
Affinity DataKi:  718nMAssay Description:Binding affinity to human BRD4 BD2 assessed as inhibition constant incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)