Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5XR8
TargetCannabinoid receptor 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582403(CHEMBL5085420)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at 3xHA tagged human CB1 receptor expressed in CHO-K1 cells assessed as reduction in forskolin-stimulated cAMP accumulation incubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Rat)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50582403(CHEMBL5085420)
Affinity DataKi:  0.390nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor assessed as inhibition constant incubated for 1 hr by TopCount scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)