Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 5Y0F
TargetFatty acid-binding protein, adipocyte(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50468371(CHEMBL4283424)
Affinity DataKi:  210nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFatty acid-binding protein, adipocyte(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50468371(CHEMBL4283424)
Affinity DataIC50: 1.69E+3nMAssay Description:Displacement of 1,8-ANS from human recombinant full length N-terminal his-tagged FABP4 expressed in Escherichia coli BL21 (DE3) incubated for 3 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFatty acid-binding protein, adipocyte(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50468371(CHEMBL4283424)
Affinity DataIC50: 1.69E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)