Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 5Y0G
TargetFatty acid-binding protein, adipocyte(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50468379(CHEMBL4295114)
Affinity DataKi:  200nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFatty acid-binding protein, adipocyte(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50468379(CHEMBL4295114)
Affinity DataKd:  1.40E+3nMAssay Description:Binding affinity to FABP4 (unknown origin) by isothermal calorimetric titration methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFatty acid-binding protein, adipocyte(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50468379(CHEMBL4295114)
Affinity DataIC50: 1.65E+3nMAssay Description:Displacement of 1,8-ANS from FABP4 (unknown origin) after 3 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)