Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5Y7K
TargetDipeptidyl peptidase 4(Human)
THE SCRIPPS RESEARCH INSTITUTE

US Patent
LigandPNGBDBM50344779((R)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: 0.300nMAssay Description:Human DPP4 activity assay data were obtained using a DPP4 Activity Assay Kit (Sigma-Aldrich, MAK088) according to the manufacturer's instructions...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2024
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
THE SCRIPPS RESEARCH INSTITUTE

US Patent
LigandPNGBDBM50344779((R)-4-((R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of recombinant human DPP-4 assessed as H-Gly-Pro-AMC cleavage after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)