Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 5Z6S
TargetPeroxisome proliferator-activated receptor gamma(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50450131(CHEMBL4164423)
Affinity DataEC50:  41nMAssay Description:Agonist activity at recombinant human GAL4-DBD fused PPARgamma LBD expressed in COS7 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50450131(CHEMBL4164423)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human Gal4-DBD fused PPARgamma LBD (unknown origin) expressed in COS-7 cells incubated for 24 hrs by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50450131(CHEMBL4164423)
Affinity DataEC50:  41nMAssay Description:Agonist activity at recombinant human GAL4-DBD fused PPARgamma LBD expressed in COS7 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)