Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 5ZK3
TargetMuscarinic acetylcholine receptor M2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H](-)-quinuclidinyl benzilate(QNB) from muscarinic (M2) receptor in rat heart homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMuscarinic acetylcholine receptor M2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PDB3D3D Structure (crystal)
TargetMuscarinic acetylcholine receptor M2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.0300nMAssay Description:Ability to displace [3H](-)-quinuclidinyl benzilate(QNB) from M2 receptor in rat heart homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMuscarinic acetylcholine receptor M2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKd:  0.200nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 using [3H]-QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)