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Report error Found 2 Enz. Inhib. hit(s) for PDB: 6E22
TargetWD repeat-containing protein 5(Human)
University of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM468882(US10807959, Example B15)
Affinity DataKd:  1.30nMAssay Description:Inhibition of human WDR5 WIN site expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetWD repeat-containing protein 5(Human)
University of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM468882(US10807959, Example B15)
Affinity DataKi:  1.33nMAssay Description:FPA Assay protocol adopted from Karatas et al. (J. Med. Chem. 2010, 5179.; J. Amer. Chem. Soc. 2013, 669.): WDR5 (Δ23, residues 24-334), is expr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)