TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Uit The Arctic University of Norway
Curated by ChEMBL
Uit The Arctic University of Norway
Curated by ChEMBL
Affinity DataKi: 2.02E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair

3D Structure (crystal)