Report error Found 4 Enz. Inhib. hit(s) for PDB: 6G27
TargetHistone-lysine N-methyltransferase NSD3(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
TargetHistone-lysine N-methyltransferase NSD3(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 6.50E+5nMAssay Description:Binding affinity to human NSD3 PWWP1 domain assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase NSD3(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 7.31E+5nMAssay Description:Binding affinity to recombinant human NSD3 PWWP1 domain (247 to 398 residues) by SPR analysisMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase NSD3(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 7.31E+5nMAssay Description:Inhibition of NSD3 PWWP1 domain (unknown origin) assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair

3D Structure (crystal)