Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 6GS6
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM139995(US8901295, F428)
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of C-terminal His6-tagged CypA (unknown origin) expressed in Escherichia coli C41(DE3) using Suc-Ala-Ala-Cis-Pro-Phe-pNA as substrate by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM139995(US8901295, F428)
Affinity DataKi:  1.68E+4nMAssay Description:Inhibition of Cyclophilin A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)