TargetHistone deacetylase 8(Blood fluke)
Martin-Luther University of Halle-Wittenberg
Curated by ChEMBL
Martin-Luther University of Halle-Wittenberg
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant Schistosoma mansoni HDAC8 expressed in Escherichia coli using Fluor de Lys as substrate preincubated for 90 mins followed b...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Blood fluke)
Martin-Luther University of Halle-Wittenberg
Curated by ChEMBL
Martin-Luther University of Halle-Wittenberg
Curated by ChEMBL
Affinity DataIC50: 191nMAssay Description:Inhibition of Schistosoma mansoni KDAC8 using (FAM)-labeled peptide as substrate after 60 mins by microfluidic assayMore data for this Ligand-Target Pair

3D Structure (crystal)