Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 6KB4
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50214899((R)-2-(3-((benzo[d]oxazol-2-yl(3-(4-methoxyphenoxy...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at Gal4-fused PPARalpha LBD (unknown origin) transfected in human HepG2 cells assessed as transcriptional activation incubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50214899((R)-2-(3-((benzo[d]oxazol-2-yl(3-(4-methoxyphenoxy...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human recombinant PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50214899((R)-2-(3-((benzo[d]oxazol-2-yl(3-(4-methoxyphenoxy...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at GAL4-tagged PPARalpha ligand-binding domain (unknown origin) expressed in HEK293T cells incubated for 16 to 19 hrs by beta-lactam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)