Report error Found 10 Enz. Inhib. hit(s) for PDB: 6M8P
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
3D Structure (crystal)TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant ERAP1 using L-leucine 7-amido-4-methyl coumarin as substrate after 5 to 10 mins by fluorescence microplate reader met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate incubated for 5 to 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant ERAP1 using L-leucine 7-amido-4-methyl coumarin as substrate after 5 to 10 mins by fluorescence microplate reader met...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant ERAP1 expressed in baculovirus infected Sf9 cells using L-leucine-7-amido-4-methyl coumarin as substrate after 5 to 1...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of ERAP1 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of wild type ERAP1 (unknown origin) using L-Rho-Succ-FKARKF as substrate preincubated for 15 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataIC50: 186nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of ERAP1 (unknown origin) using L-AMC as substrateMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Wroclaw University of Technology
Curated by ChEMBL
Wroclaw University of Technology
Curated by ChEMBL
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of human ERAP1More data for this Ligand-Target Pair