Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 6O1S
TargetPlasma kallikrein(Human)
Novartis

US Patent
LigandPNGBDBM212113(US9290485, 145)
Affinity DataIC50: 0.200nMpH: 7.8 T: 2°CAssay Description:Enzymatic reactions were conducted in assay buffer , comprising 50 mM Hepes/NaOH at pH 7.8, 150 mM NaCl, 1 mM EDTA and 0.05% (w/v) CHAPS. For the det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2017
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetPlasma kallikrein(Human)
Novartis

US Patent
LigandPNGBDBM212113(US9290485, 145)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human plasma kallikrein incubated for 1 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)