Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 6PNO
TargetGlutathione S-transferase omega-1(Human)
Monash University

Curated by ChEMBL
LigandPNGBDBM50527184(CHEMBL4454026)
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutathione S-transferase omega-1(Human)
Monash University

Curated by ChEMBL
LigandPNGBDBM50527184(CHEMBL4454026)
Affinity DataKi:  4.80E+3nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli assessed as inhibitor constant using S-(4-nitrophenacyl)glutathione ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)