Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 6Q3Y
TargetBromodomain-containing protein 4(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50526295(CHEMBL4469087)
Affinity DataKd:  54nMAssay Description:Binding affinity to BRD4 (unknown origin) by isothermal calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50526295(CHEMBL4469087)
Affinity DataIC50: 540nMAssay Description:Inhibition of full-length C-terminal NanoLuc-tagged BRD4 BD1 (unknown origin) expressed in human HEK293 cells after 2 hrs by NanoBRET target engageme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)