Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) for PDB: 6QBA
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50019040(CHEMBL1230001)
Affinity DataIC50: 0.155nMAssay Description:Antagonist activity at maltose binding protein-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as inhibition of retinol-induced p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50019040(CHEMBL1230001)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant RBP4-transthyretin interaction by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50019040(CHEMBL1230001)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]-retinol from RBP4 (unknown origin) by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50019040(CHEMBL1230001)
Affinity DataIC50: 15nMAssay Description:Competitive displacement of 3[H]retinol from biotinylated RBP4 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50019040(CHEMBL1230001)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]retinol from biotinylated human RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50019040(CHEMBL1230001)
Affinity DataIC50: 89nMAssay Description:Displacement of [3H]-retinol from human recombinant RBP4 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinol-binding protein 4(Human)
Albany Molecular Research

Curated by ChEMBL
LigandPNGBDBM50019040(CHEMBL1230001)
Affinity DataIC50: 122nMAssay Description:Inhibition of retinol-induced interaction of bacterially expressed MBP-tagged RBP4 (unknown origin) with Eu3+ cryptate labeled TTR by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)