Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 6RWJ
TargetBromodomain-containing protein 4(Human)
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559313(CHEMBL4783790)
Affinity DataKd:  641nMAssay Description:Binding affinity to BRD4 bromo domain 1 (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559313(CHEMBL4783790)
Affinity DataKd:  6.41E+3nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 25 degree C by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)