Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 6SA2
TargetBromodomain-containing protein 4(Human)
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559309(CHEMBL4762147)
Affinity DataKd:  80nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 25 degree C by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559309(CHEMBL4762147)
Affinity DataKd:  60nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)