Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 6U0D
TargetBromodomain-containing protein 4(Human)
Md Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50584382(CHEMBL5090401)
Affinity DataIC50: 90nMAssay Description:Binding affinity recombinant human BRD4 BD1 (42 to 168 residues) expressed in Escherichia coli BL21(DE3) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
Md Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50584382(CHEMBL5090401)
Affinity DataIC50: 1.09E+3nMAssay Description:Binding affinity human BRD4 BD2 incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)