Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 6VYJ
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50608079(CHEMBL5286019)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50608079(CHEMBL5286019)
Affinity DataEC50:  2.90E+4nMAssay Description:Inhibition of His tagged UHRF1 tandem Tudor domain (unknown origin) using biotinylated-H3K9me3 peptide as substrate incubated for 1 hr by TR-FRET ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetE3 ubiquitin-protein ligase UHRF1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50608079(CHEMBL5286019)
Affinity DataEC50:  2.92E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMedPDB3D3D Structure (crystal)