Affinity DataIC50: 200nMAssay Description:Binding affinity to BRD9 (unknown origin) N-terminal bromodomain by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity to human partial length BRD9 (R130 to V259 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair

3D Structure (crystal)