Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 6YUM
TargetCasein kinase II subunit alpha(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50556137(CHEMBL4793819)
Affinity DataIC50: 8nMAssay Description:Displacement of fluorescent tracer from full-length human C-terminal NanoLuc-tagged CK2alpha expressed in HEK293T permeabilized cells measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50556137(CHEMBL4793819)
Affinity DataIC50: 8nMAssay Description:Inhibition of CK2alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50556137(CHEMBL4793819)
Affinity DataKd:  12nMAssay Description:Binding affinity to N-terminal His6-tagged CK2alpha (1 to 337 residues) (unknown origin) expressed in BL21(DE3) cells by isothermal titration calorim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50556137(CHEMBL4793819)
Affinity DataIC50: 1.51E+3nMAssay Description:Displacement of fluorescent tracer from full-length human C-terminal NanoLuc-tagged CK2alpha expressed in HEK293T cells measured after 2 hrs by NanoB...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)