Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) for PDB: 7JSJ
TargetSolute carrier family 13 member 5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149294(CHEMBL3769578)
Affinity DataIC50: 501nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 13 member 5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149294(CHEMBL3769578)
Affinity DataIC50: 501nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 13 member 5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149294(CHEMBL3769578)
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 13 member 5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149294(CHEMBL3769578)
Affinity DataIC50: 1.62E+4nMAssay Description:Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 13 member 5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149294(CHEMBL3769578)
Affinity DataIC50: 1.62E+4nMAssay Description:Inhibition of SLC13A5 in human hepatocyte cells assessed as reduction in citrate uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMedPDB3D3D Structure (crystal)