Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 7LPK
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573183(CHEMBL4867912)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
Fujian Medical University

Curated by ChEMBL
LigandPNGBDBM50573183(CHEMBL4867912)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)