Report error Found 2 Enz. Inhib. hit(s) for PDB: 7LUK
Affinity DataEC50: 2.5nMAssay Description:Inverse agonist activity at human Gal4-fused RORgammat expressed in human Jurkat cells luciferase reporter gene assayMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataEC50: 26nMAssay Description:Inverse agonist activity at RORgammat in human whole blood assessed as inhibition of anti-CD3/anti-CD28 monoclonal antibodies-stimulated IL-17A produ...More data for this Ligand-Target Pair