Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 7TUZ
TargetG-protein coupled receptor 183(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50558426(CHEMBL4788348)
Affinity DataEC50:  0.0320nMAssay Description:Agonist activity at Go2-q-coupled human EBI2 expressed in COS7 cell membranes assessed as stimulation of [35S]GTPgammaS binding preincubated for 20 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetG-protein coupled receptor 183(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50558426(CHEMBL4788348)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at Go2-q-coupled EBI2 (unknown origin) expressed in COS7 cell membranes assessed as stimulation of [35S]GTPgammaS binding preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetG-protein coupled receptor 183(Mouse)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50558426(CHEMBL4788348)
Affinity DataEC50:  0.702nMAssay Description:Agonist activity at Go2-q-coupled mouse EBI2 expressed in COS7 cell membranes assessed as stimulation of [35S]GTPgammaS binding preincubated for 20 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetG-protein coupled receptor 183(Rat)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50558426(CHEMBL4788348)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at Go2-q-coupled rat EBI2 expressed in COS7 cell membranes assessed as stimulation of [35S]GTPgammaS binding preincubated for 20 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)