Compile Data Set for Download or QSAR
Report error Found 1 Enz. Inhib. hit(s) for PDB: 7VUI
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50132143(CHEMBL3633720)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)