Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 7W0G
TargetPeroxisome proliferator-activated receptor delta(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50584465(CHEMBL5084377)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at human PPARdelta transfected in Cos7 cells co-expressing with pBIND and pGL4.35 Gal4 UAS Luc reporter plasmid by measuring lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50584465(CHEMBL5084377)
Affinity DataEC50:  8.40nMAssay Description:Agonist activity at PPARdelta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50584465(CHEMBL5084377)
Affinity DataEC50:  9.70nMAssay Description:Agonist activity at human PPARdelta transfected in african green monkey COS7 cells assessed transactivation incubated for 16 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50584465(CHEMBL5084377)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse PPARdelta in Cos7 cells transfected with pBIND and pGL4.35 Gal4 UAS Luc reporter plasmid by measuring luciferase activity i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)