Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) for PDB: 7WGL
TargetPeroxisome proliferator-activated receptor delta(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28701(Cedur | 2-(4-{2-[(4-chlorophenyl)formamido]ethyl}p...)
Affinity DataEC50:  1.89E+4nMAssay Description:Agonist activity at human PPARdelta expressed in HepG2 cells co-transfected with PPRE3-TK-luc assessed as beta-galactosidase activity after 20 to 22 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28701(Cedur | 2-(4-{2-[(4-chlorophenyl)formamido]ethyl}p...)
Affinity DataEC50:  2.00E+4nMAssay Description:Compound was tested for agonist activity on human Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28701(Cedur | 2-(4-{2-[(4-chlorophenyl)formamido]ethyl}p...)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity for Human PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28701(Cedur | 2-(4-{2-[(4-chlorophenyl)formamido]ethyl}p...)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at human PPARdelta expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28701(Cedur | 2-(4-{2-[(4-chlorophenyl)formamido]ethyl}p...)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at human PPARdelta expressed in monkey CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28701(Cedur | 2-(4-{2-[(4-chlorophenyl)formamido]ethyl}p...)
Affinity DataEC50:  3.57E+4nMAssay Description:Agonist activity at human PPARdelta expressed in HEK293 cells cotransfected with PPREx4-TK-luc assessed as activation of luciferase activity measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28701(Cedur | 2-(4-{2-[(4-chlorophenyl)formamido]ethyl}p...)
Affinity DataEC50:  1.02E+5nMAssay Description:In vitro transcriptional activation of hPPAR deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM28701(Cedur | 2-(4-{2-[(4-chlorophenyl)formamido]ethyl}p...)
Affinity DataEC50:  1.10E+5nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor delta-GAL4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM28701(Cedur | 2-(4-{2-[(4-chlorophenyl)formamido]ethyl}p...)
Affinity DataEC50:  1.10E+5nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28701(Cedur | 2-(4-{2-[(4-chlorophenyl)formamido]ethyl}p...)
Affinity DataEC50: >1.43E+5nMAssay Description:Agonist activity on Gal4 chimeric human Peroxisome proliferator activated receptor delta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)