Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 7Z4U
TargetYTH domain-containing family protein 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50601386(CHEMBL5201513)
Affinity DataIC50: 1.61E+5nMAssay Description:Inhibition of YTHDF2 YTH domain (unknown origin) (383 to 579 residues) expressed as Escherichia coli BL21 (DE3) Rosetta cells by HTFR based binding a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetYTH domain-containing family protein 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50601386(CHEMBL5201513)
Affinity DataIC50: 4.91E+5nMAssay Description:Binding affinity to GST-tagged YTHDF2 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)